Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04886
Ion Channel
Sodium channel protein type 9 subunit alpha
Peptide Function
Inhibitor
Gene Name
SCN9A
Activity Data (nM)
IC50
13 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
DCLGAMRKCIPDNDKCCRPNLVCSRTHKWCKYVF
Peptide UniProt Accession
Not available
UniParc
UPI0003E5FFFF
Peptide Synonyms/Alias
[CHEMBL3416893; BDBM50077464]
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
Not available
Experimental Conditions
pH
Extracellular solution: pH 7.4/Intracellular solution: pH 7.3
Holding Potential (mV)
−125 to −10 mV
Temperature
~22 °C
Test Method
Patch-clamping
Test Species
Not specified
Binding Information
Binding Site
Extracellular domain
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Mus musculus (Mouse)
References & Disease Information
Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available